Sunday, 8 April 2012

Estradiol Gel Packets



Pronunciation: ES-tra-DYE-ol
Generic Name: Estradiol
Brand Name: Divigel

Estradiol Gel Packets should not be used to prevent heart disease, heart attacks, strokes, or dementia. Estrogens have been shown to increase the risk of heart disease (including heart attack), stroke, dementia, serious blood clots (eg, in the lungs or legs), cancer of the uterus, and breast cancer in some women. Tell your doctor right away if you have unusual vaginal bleeding while you use Estradiol Gel Packets. Talk with your doctor if you have questions about the benefits and risks of using Estradiol Gel Packets.


Estradiol Gel Packets should be used for the shortest possible time at the lowest effective dose to minimize the risk of these side effects. Talk with your doctor regularly about your need to use Estradiol Gel Packets.





Estradiol Gel Packets are used for:

Treating certain moderate to severe symptoms of menopause (eg, hot flashes).


Estradiol Gel Packets are an estrogen hormone. It works by replacing estrogen in the body when it no longer produces enough on its own.


Do NOT use Estradiol Gel Packets if:


  • you are allergic to any ingredient in Estradiol Gel Packets

  • you are pregnant or suspect you may be pregnant

  • you have undiagnosed abnormal vaginal bleeding

  • you have a history of blood clots (eg, in the lungs, legs, eyes); endometrial, cervical, or vaginal cancer; estrogen-dependent growths; breast cancer; or liver problems

  • you have had a heart attack or stroke within the past 12 months

Contact your doctor or health care provider right away if any of these apply to you.



Before using Estradiol Gel Packets:


Some medical conditions may interact with Estradiol Gel Packets. Tell your doctor or pharmacist if you have any medical conditions, especially if any of the following apply to you:


  • if you are pregnant, planning to become pregnant, or are breast-feeding

  • if you are taking any prescription or nonprescription medicine, herbal preparation, or dietary supplement

  • if you have allergies to medicines, foods, or other substances

  • if you have a history of endometriosis, growths in the uterus, abnormal mammogram, abnormal vaginal bleeding, a lump in the breast, or fibrocystic breast disease, or if a family member has had breast cancer

  • if you have dementia or other memory problems, or abnormal blood calcium levels

  • if you have a history of asthma, cancer, high blood cholesterol or lipid levels, diabetes, heart problems, high blood pressure, heart attack or stroke, kidney problems, liver tumor, mental or mood problems (eg, depression), underactive thyroid, migraine headaches, gallbladder or pancreas problems, seizures (eg, epilepsy), lupus, chorea, or the blood disease porphyria

  • if you smoke, are very overweight, or will be having surgery

  • if you have a history of yellowing of the eyes or skin during pregnancy or with past estrogen use

  • if a member of your family has a history of blood clots (eg, in the legs, lungs, eyes), diabetes, lupus, or obesity

  • if you have had your uterus removed (hysterectomy)

Some MEDICINES MAY INTERACT with Estradiol Gel Packets. Tell your health care provider if you are taking any other medicines, especially any of the following:


  • Azole antifungals (eg, ketoconazole), HIV protease inhibitors (eg, ritonavir), or macrolide antibiotics (eg, erythromycin) because they may increase the risk of Estradiol Gel Packets's side effects

  • Barbiturates (eg, phenobarbital), carbamazepine, hydantoins (eg, phenytoin), rifampin, or St. John's wort because they may decrease Estradiol Gel Packets's effectiveness

  • Thyroid hormones (eg, levothyroxine) because their effectiveness may be decreased by Estradiol Gel Packets

This may not be a complete list of all interactions that may occur. Ask your health care provider if Estradiol Gel Packets may interact with other medicines that you take. Check with your health care provider before you start, stop, or change the dose of any medicine.


How to use Estradiol Gel Packets:


Use Estradiol Gel Packets as directed by your doctor. Check the label on the medicine for exact dosing instructions.


  • An extra patient leaflet is available with Estradiol Gel Packets. Talk to your pharmacist if you have questions about this information.

  • Apply Estradiol Gel Packets to the upper thigh area of the right or left leg. Change between your left and right thigh each day to help avoid skin irritation.

  • Apply Estradiol Gel Packets to clean, intact skin only. Be sure the area is completely dry before applying Estradiol Gel Packets.

  • Do not apply Estradiol Gel Packets to skin that is irritated or broken. Do not apply it to your face, in or around the vagina, or to your breasts.

  • If you take a bath or shower, or use a sauna around the time of your dose, apply Estradiol Gel Packets afterwards. Be sure the area is completely dry before applying the medicine.

  • Open the packet and squeeze the entire contents of the packet onto the upper thigh of one leg. Gently spread the medicine as thinly as possible over an area of about 5 to 7 inches (about 2 palm prints). You do not need to rub the medicine in.

  • Throw away the empty packet in the trash out of the reach of children and pets.

  • Wash your hands with soap and water after using Estradiol Gel Packets.

  • Cover the application site with clothing after the medicine is completely dry. This will help to prevent others from coming into contact with the medicine. Be sure the medicine is completely dry before you dress.

  • Do not wash the application site for at least 1 hour after you apply Estradiol Gel Packets.

  • Do not allow others to apply Estradiol Gel Packets for you. Do not allow others to come into contact with the application site for at least 1 hour after you apply Estradiol Gel Packets. If someone else comes into contact with Estradiol Gel Packets, have them wash the area with soap and water right away.

  • Use Estradiol Gel Packets at the same time each day.

  • If you spill some of Estradiol Gel Packets while you are applying it, do not open a new packet. Wait and apply your regular dose the next day.

  • If you miss a dose of Estradiol Gel Packets, use it as soon as possible. If your next dose is less than 12 hours away, skip the missed dose and go back to your regular dosing schedule. Do not use 2 doses at once.

Ask your health care provider any questions you may have about how to use Estradiol Gel Packets.



Important safety information:


  • Estradiol Gel Packets are for external use only. Do not get it in your eyes, nose, vagina, or mouth. If you get it in any of these areas, rinse right away with warm clean water.

  • Check with your doctor before applying sunscreen to the application site while using Estradiol Gel Packets.

  • If you will be swimming, wait until Estradiol Gel Packets are completely dry before going into the water.

  • Estradiol Gel Packets are flammable. Avoid fire, flame, or smoking until the medicine has dried on your skin.

  • Eating grapefruit or drinking grapefruit juice may increase the risk of Estradiol Gel Packets's side effects. Talk to your doctor before including grapefruit or grapefruit juice in your diet while you are taking Estradiol Gel Packets.

  • Tell your doctor or dentist that you take Estradiol Gel Packets before you receive any medical or dental care, emergency care, or surgery. If possible, Estradiol Gel Packets should be stopped at least 4 to 6 weeks before surgery or any time you might be confined to a bed or chair for a long period of time (such as a long plane flight, car ride, bedrest, or illness).

  • Estradiol Gel Packets may cause dark skin patches on your face. Exposure to the sun may make these patches darker. If patches develop, use a sunscreen or wear protective clothing when exposed to the sun, sunlamps, or tanning booths.

  • If you wear contact lenses and you develop problems with them, contact your doctor.

  • Diabetes patients - Estradiol Gel Packets may affect your blood sugar. Check blood sugar levels closely. Ask your doctor before you change the dose of your diabetes medicine.

  • Estradiol Gel Packets may interfere with certain lab tests. Be sure your doctor and lab personnel know you are using Estradiol Gel Packets.

  • Lab tests and medical exams, including breast exams, mammograms, Pap tests, physicals, and blood pressure, may be performed while you use Estradiol Gel Packets. These tests may be used to monitor your condition or check for side effects. Be sure to keep all doctor and lab appointments.

  • Examine your breasts monthly as directed by your doctor. Report any lumps right away.

  • Estradiol Gel Packets should not be used in CHILDREN; safety and effectiveness in children have not been confirmed.

  • PREGNANCY and BREAST-FEEDING: Do not use Estradiol Gel Packets if you are pregnant. If you think you may be pregnant, contact your doctor right away. Estradiol Gel Packets are found in breast milk. If you are or will be breast-feeding while you use Estradiol Gel Packets, check with your doctor. Discuss any possible risks to your baby.


Possible side effects of Estradiol Gel Packets:


All medicines may cause side effects, but many people have no, or minor, side effects. Check with your doctor if any of these most COMMON side effects persist or become bothersome:



Breast pain or tenderness; headache; mild hair loss; mild nausea or vomiting; spotting or breakthrough bleeding; stomach cramps or bloating.



Seek medical attention right away if any of these SEVERE side effects occur:

Severe allergic reactions (rash; hives; itching; difficulty breathing; tightness in the chest; swelling of the mouth, face, lips, or tongue; unusual hoarseness); blurred or double vision, vision loss, or other vision changes; breast lump or discharge; calf or leg pain or swelling; chest pain; confusion; coughing up blood; fainting; memory problems; mental or mood changes (eg, depression); migraine headache; numbness of an arm or leg; one-sided weakness; persistent or recurring abnormal vaginal bleeding; severe or persistent headache or dizziness; severe or persistent stomach pain, nausea, or vomiting; shortness of breath; slurred speech; swelling of the hands, legs, or feet; vaginal discharge, itching, or odor; yellowing of the skin or eyes.



This is not a complete list of all side effects that may occur. If you have questions about side effects, contact your health care provider. Call your doctor for medical advice about side effects. To report side effects to the appropriate agency, please read the Guide to Reporting Problems to FDA.



If OVERDOSE is suspected:


Contact 1-800-222-1222 (the American Association of Poison Control Centers), your local poison control center, or emergency room immediately. Symptoms may include abnormal vaginal bleeding; or severe or persistent nausea or vomiting.


Proper storage of Estradiol Gel Packets:

Store Estradiol Gel Packets at room temperature, between 68 and 77 degrees F (20 and 25 degrees C) with the cap secured. Brief storage at temperatures between 59 and 86 degrees F (15 and 30 degrees C) is permitted. Store away from heat, moisture, and light. Do not store in the bathroom. Keep Estradiol Gel Packets out of the reach of children and away from pets.


General information:


  • If you have any questions about Estradiol Gel Packets, please talk with your doctor, pharmacist, or other health care provider.

  • Estradiol Gel Packets are to be used only by the patient for whom it is prescribed. Do not share it with other people.

  • If your symptoms do not improve or if they become worse, check with your doctor.

  • Check with your pharmacist about how to dispose of unused medicine.

This information is a summary only. It does not contain all information about Estradiol Gel Packets. If you have questions about the medicine you are taking or would like more information, check with your doctor, pharmacist, or other health care provider.



Issue Date: February 1, 2012

Database Edition 12.1.1.002

Copyright © 2012 Wolters Kluwer Health, Inc.

More Estradiol resources


  • Estradiol Use in Pregnancy & Breastfeeding
  • Drug Images
  • Estradiol Drug Interactions
  • Estradiol Support Group
  • 57 Reviews for Estradiol - Add your own review/rating


Compare Estradiol with other medications


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  • Breast Cancer, Palliative
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  • Oophorectomy
  • Osteoporosis
  • Postmenopausal Symptoms
  • Primary Ovarian Failure
  • Prostate Cancer

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